Page 46 - CW E-Magazine (9-7-2024)
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PHARMACEUTICAL ADVANCED INTERMEDIATES                                                                                         Available following material with us regularly


                PRODUCT NAMES      CAS No  PHARMACEUTICAL        PRODUCT NAMES      CAS No  PHARMACEUTICAL
                                            INTERMEDIATES                                    INTERMEDIATES
        1-(1-Ethoxyethyl)-1H-pyrazole-4-boronic acid   1029716-44-6 Ruxolitinib/Baricitinib  4-Fluorophenylboronic Acid  1765-93-1  Canagliflozin
        pinacol ester                                    4-Formylphenylboronic acid  87199-17-5  Atazanavir/Rucaparib
        1-(Tetrahydro-2H-pyran-2-yl)-1H-pyrazole-5-boronic 903550-26-5 Asciminb  4-Methoxy-5-(3-morpholino propoxy)-2-nitroben-  675126-26-8 Gefitinib
        acid pinacol ester                               zonitrile                                                                  DIMETHYL FORMAMIDE
        1-Isopropylpyrazole-5-boronic acid pinacol ester  1282518-60-8 Voxelotor  4-Phenoxybenzoic acid  2215-77-2  Ibrutinib
        1-Methylpyrazole-4-boronic acid pinacol ester  761446-44-0 Ruxolitinib/Baricitinib /   4-Phenoxyphenylboronic acid  51067-38-0  Ibrutinib / Tolebrutinib
                                         Avatrompobag / Savolitinib /                                                                            – CHEMANOL., SAUDI ARABIA
                                         Erdafitinib     4-Pyrazoleboronic acid pinacol ester  269410-08-4 Ruxolitinib
        1-Phenyl-5-pyridin-2-ylpyridin-2-one  381725-50-4 Perampanel  4-Tolylboronic acid  08-05-5720  Olmesartan/Zibotentan
        2-(4-Fluorophenyl)thiophene  58861-48-6  Canagliflozin  4,4’-Dimethoxybenzil   1226-42-2  Flumizole/Idanpramine
        2-(5-Bromo-2-methylbenzyl)-5-(4-fluorophenyl)  1030825-20-7 Canagliflozin  4,5-Dimethoxy-1-cyanobenzocyclobutane  35202-54-1  Ivabradine
        thiophene                                        4,6-Dichloro-2-methyl pyrimidine  1780-26-3  Dasatanib
        2-Acetyl-4-chlorothiophene  34730-20-6  Avatrompobag  5-(2-Pyridyl)-1,2-dihydro pyridine-2-one  381233-78-9 Perampanel  • 1, 4 Butanediol       • DL Tartaric Acid           • N-Heptane 99%
        2-Bromo-4’-cyanoacetophenone  20099-89-2  Isavuconazole  5-Acetylthiophene-2-carboxylic acid  4066-41-5  Arotinolo HCL  • 1-Bromo-3-Chloropropane   • EDTA 2Na               • N Hexane 99%
        2-Bromoethylamine hydrobromide  2576-47-8  Altanserin/Medazepam  5-Aminoisoquinoline  1125-60-6  Taprizosin
        2-Chloro-4,6-dimethoxy-1,3,5-triazine  3140-73-6  Pemetrexid  5-Bromo-2-methylbenzoic acid  79669-49-1  Canagliflozin  • 2 Ethyl Hexyl Acrylate  • Epichlorohydrine          • N Propanol
        2-Chloro-5-Nitrophenylboronic acid  867333-29-7 Zanubritinib  5-Chlorothiophene-2-carboxylic acid  24065-33-6  Rivaroxaban  • 2 Hydroxy Propyl Methacrylate (2HPMA) • Ethyl Aceto Acetate  • Neo Pentyl Glycol
        2-Cyanophenylboronic acid 1,3-propanediol Ester  172732-52-4 Perampanel  5-Formyl-2-furylboronic acid  27329-70-0  Lapatinib  • 2 Methyl Tetra Hydro Furan   • Ethyl Acrylate   • Nonyl Phenol
        2-Fluorophenylboronic acid.   01993-03-9  Vonoprazan.   5-Formyl-2,4-dimethyl-1H-pyrrole-3-carboxylic acid 253870-02-9 Sunitinib  • 2, 2-Dimethoxy Propane   • Ethyl Chloro Formate  • Para Tertiary Butyl Phenol
        2-Fluoro-3-Methoxyphenyl boronic Acid  352303-67-4 Elagolix  5-Methyl-2-(2H-1,2,3-triazol-2-yl)benzoic acid  956317-36-5 Suvorexant
        2-Formylphenylboronic acid  40138-16-7  Perampanel  6-(Dimethylamino)quinaldine  92-99-9  Pyrvinium(Viprynium)  • 2-Ethyl Hexanoic Acid         • Ethyl Cyano Acetate        • Paraformaldehyde 91%
        2-Methoxypyridine-5-boronic acid  163105-89-3 Perampanel  6-Bromo-2-tetralone  4133-35-1  Izonstride            • 2-Hydroxy Ethyl Acrylate (2-HEA)   • Ethylene Diamine      • Paraformaldehyde 96%
        2-Tolylboronic acid                                                          16419-60-6  Befetupitant/Natupitant  6-Bromopyridine-3-carbaldehyde  149806-06-4 Abemaciclib  • 2-Hydroxy Propyl Acrylate (2-HPA)  • Formic Acid 99%  • Piperazine Anhydrous
        2,3-Dimethyl-2H-indazol-6-amine Hydrochloride  635702-60-2 Pazopanib   7-Methoxy-6-(3-morpholin-4-ylpropoxy)-1H-  199327-61-2 Gefitinib  • 2-Hydroxyethyl Methacrylate (HEMA)   • Hexylene Glycol   • Poly Propylene Glycol 1000
        2,3-Dimethylindazol-6-amine  444731-72-0 Pazopanib  quinazolin-4-one
        2,4-Difluorophenylboronic acid  144025-03-6 Diflunisal  Alpha-Bromo-gama-butyrolactone  5061-21-2  Delgocitinib  • 2-Methyl-1, 3-Propanediol    • Hydroquinone               • Poly Propylene Glycol 2000
        3-(Hydroxymethyl)phenyl boronic acid  87199-15-3  Fasigliflam,Pacritinib  Anisaldehyde dimethyl acetal  2186-92-7  Roxaticin  • Acrylamide      • Hydroxylamine Hydrochloride    • Poly Propylene Glycol 400
        3-Amino-4-methyl thiophehne-2-carboxylic acid  85006-31-1  Articaine  Benzaldehyde dimethyl acetal  1125-88-8  Fondaparinux Sodium/     • Acrylic Acid   (Drum Packing)      • Potassium Carbonate Granular
                                                                                          Mifamurtide/Minamyl
        3-Aminophenylacetylene   54060-30-9  Erlotinib/Solithromycin                      tripeptide                    • Adipic Acid                   • Hydroxylamine Sulfate      • Potassium Carbonate Powder
        3-Bromo-1-phenyl-5-pyridin-2-ylpyridin-2-one  381248-06-2 Perampanel  Ethyl 5-bromobenzofuran-2-carboxylate  84102-69-2  Vilazodone             • Iso Butyric Acid
        3-Bromobenzyl cyanide    31938-07-5  Bimosiamose/Bioresmethrin  Ethyl N-[(3,4-dimethoxy-7-bicyclo[4.2.0]  148870-55-7 Ivabradine  • Allyl Chloride                           • Propionaldehyde
        3-Bromoquinoline         5332-24-1  Tariquidar   octa-1,3,5-trienyl)methyl]carbamate                            • Amino Ethyl Ethanolamine (AEEA)   • Isophthalic Acid       • Propionic Acid
        3-Carboxyphenylboronic acid  25487-66-5  Eltrombopag  Isobutylboronic Acid  84110-40-7  Bortezomib/Ixazomib Cytrate   • Benzoic Acid            • Isovaleraldehyde           • Propylene Carbonate
        3-Chlorophenylboronic acid  63503-60-6  Vadadustat  Isopropoxyboronic acid pinacol ester  61676-62-8  Ruxolitinib/Baricitinib  • Butyl Glycol   • L + Tartaric Acid          • Propylene Glycol Mono Methyl Ether
        3-Fluorophenylboronic acid  768-35-4  Vorapaxar / Polmacoxib  Methoxyboronic acid pinacol ester   1195-66-0  Crizotinib                         • Maleic Anhydride
        3-Formylphenylboronicacid  87199-16-4  Fasigliflam  Triethyloxonium Tetrafluoroborate  368-39-8  Fezolinetant   • Caustic Potash                                             • Propylene Glycol Monomethylether Acetate
        3-Iodo-1H-pyrazolo[3,4-d] pyrimidin-4-amine  151266-23-8 Ibrutinib  Methyl 1-((4-fluorophenyl) carbamoyl) cyclopro-  1345847-71-3 Cabozantinib  • D – Tartaric Acid  • MDI (Cosmonate M-200)   • Propylene Glycol Tech
                                                         pane carboxylate
        3-Tolylboronic acid                                                              17933-03-8  Eltrombopag  N-Acetyl-2-cyanoglycine ethyl ester  4977-62-2  Cetrorelix/Lanreotide  • Di Basic Ester  • Methacrylic Acid  • Propylene Glycol USP
        4-(2-Pyridinyl)benzaldehyde  127406-56-8 Atazanavir  N-Boc -Pyrrole       5176-27-2  Tanaproget                 • Di Iso Propyl Ether           • Methane Sulphonic Acid     • Sodium Borohydride Powder
        4-(3-Fluorophenyl)-2,2-dimethyl-5-(4-(methyl   301693-70-9 Polmacoxib  N-Boc-2-pyrroleboronic Acid  135884-31-0 Tanaproget
        sulfinyl)phenyl)furan-3(2H)-one                                                                                 • Di N Butylamine               • Methyl Acrylate            • Sodium Citrate
        4-(Benzyloxycarbonylamino)-2-fluorophenylboronic  874290-59-2 Tedizolid  N-Boc-ethanolamine  26690-80-2  Indinavir/Brostacillin  • Di Propylene Glycol [Industrial Grade]  • Methyl Cyano Acetate   • Sodium Gluconate
        acid                                             N-Pyridin-2-yl-4-(4,4,5,5-tetramethyl-[1,3,2]dioxa  1383385-64-5 Acalabrutinib
        4-(Bromomethyl)phenylboronic acid pinacol ester 138500-85-3 Filgotinib  borolan-2-yl)-benzamide                 • Di Propylene Glycol FrG Grade   • Methyl Cyclohexane       • Sodium Metal
        4-(Hydroxymethyl)phenylboronic acid  59016-93-2  Filgotinib  Phenylboronic acid  98-80-6  Perampanel/ Eslicar-  • Dicyandiamide                 • Methyl Methacrylate        • Succinic Acid
                                                                                          bazepine / Vofopitant
        4-(Pyridin-2-ylcarbamoyl) phenylboronicacid  850568-25-1 Acalabrutinib            Cis-Losofoxifene / Simvastatin            • Diethanolamine    • Methyl Propyl Ketone       • Tert-Butylamine
        4-Bromo-1-(1-ethoxyethyl)-1H-pyrazole  1024120-52-2 Ruxolitinib/Baricitinib  Pyridine-3-boronic Acid  1692-25-7  Aberiterone/Niraparib  • Diethyl Malonate  • Methyl Tertiary Butyl Ether  • Tertiary Butanol
        4-Bromophenylboronic acid  5667-74-3  Aprocitentan  Pyridine-4-boronic acid  1692-15-5  Ceritinib/ Tirofiban Hydro-
        4-Bromopyrazole          2075-45-8  Ruxolitinib/Baricitinib                       chloride                      • Dimethyl Acetamide            • Mono Iso Propylamine 70%   • Tetra Hydro Furan
        4-Carboxyphenylboronic acid  14047-29-1  Lumacaftor/Zibotentan  Tri-o-tolylphosphine  6163-58-2  Eletripatan/Rilpivirine  • Dimethyl Formamide  • Mono-N-Butylamine          • Toluene Di Isocyanate
        4-Chloro-7H-pyrrolo[2,3-d]pyrimidine  3680-69-1  Ruxolitinib/Baricitinib  Tri-tert-butyl phosphonium tetrafluoroborate  131274-22-1 Lumacaftor  • Dimethyl Malonate  • Morpholine   • Tri Ethyl Ortho Formate
        4-Chlorophenylboronic acid  1679-18-1  Boscalid / Vemurafenib  Trimethyloxonium tetrafluoro borate  420-37-1  Dolastatin/Ertapenem/Imipen-  • Dimethyl Sulfoxide   • N Butyl Methacrylate  • Tri Methyl Ortho Formate
                                                                                          em/Sitagliptin/Pazopanib
                                                                                                                        • Dipropylene Glycol Mono Methyl Ether  • N Butyraldehyde    • Tri Methylol Propane
                                                                                                                                                  Contact us for your requirements:
                                                                                                                                                  Leo Chemo Plast Pvt. Ltd.
                            DENISCO CHEMICALS PVT. LTD                                                                                            B / 126, Ghatkopar Industrial Estate, Off. LBs Marg,
                                                                                                                                                  Behind R City Mall, Ghatkopar (W), Mumbai - 400 086.
                       Plot 1040, Road 51, Jubilee Hills - 500033. Hyderabad (Telangana) INDIA.                                                   Board Line : 022-35230401 / 35230260 / 35153967 / 35014906
                                   Off: (91-40) 23552990 w Mob: (91) 9989050754                                                                   Email: info@leochemo.com w Visit us at: www.leochemo.com
                                  Email: products@denisco.com w www.denisco.com

       46                                                                        Chemical Weekly  July 9, 2024


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